发明名称 ALPHA ANOMER ENRICHED MIXTURE OF 3,5-BIS (PROTECTED HYDROXY)-2-DEOXY-2,2-DIFLUORO-D-RIBOFURANOSYL-1-ALKYL-(ORARYL)-SULFONATES AND THEIR PREPARATION AT LOW TEMPERATURES
摘要 <p>A stereoselective process for preparing alpha-anomer enriched 2-deoxy-2,2-difluoro-D-ribofuranosyl sulfonates by contacting a lactol with an base in an inert solvent, adjusting the temperature and adding a sulfonating reagent.</p>
申请公布号 IL106076(A) 申请公布日期 2002.02.10
申请号 IL19930106076 申请日期 1993.06.21
申请人 ELI LILLY AND COMPANY 发明人
分类号 C07H11/00;C07H13/08;(IPC1-7):C07H13/00 主分类号 C07H11/00
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