发明名称 METHOD FOR THE SEPARATION OF INTERMEDIATES WHICH MAY BE USED FOR THE PREPARATION OF ESCITALOPRAM
摘要 The present invention relates to a novel method for the preparation of diol intermediates having the formula (II) and/or the opposite enantiomer of an acylated diol having the formula (IV) useful for the preparation of escitalopram involving selective enzymatic acylation or deacylation.
申请公布号 MEP1608(A) 申请公布日期 2010.02.10
申请号 MEP1608 申请日期 2003.08.12
申请人 H.LUNDBECK A/S 发明人 TAOKA NAOAKI;KATO TAKAHISA;YAMAMOTO SHOGO;YOSHIDA TAKASHI;TAKEDA TOSHIHIRO;UEDA YASUYOSHI;PETERSEN HANS;DANCER ROBERT;AHMADIAN HALEH;LYNGSOE LARS OLE
分类号 C12P13/00;C07B57/00;C07C253/30;C07C253/34;C07C255/34;C07C255/53;C07C255/59;C07D307/87 主分类号 C12P13/00
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