| 摘要 |
Benzothiazine derivs. of general formula I and their dehydration and redn. products and acid addn. and quaternary ammonium salts. Y = S, SO ro SO2 X and X' = OH, Alkyl, alkoxy, aryloxy, alkylthio, NO2, NH2, Hal or CF3. Preferred are H and Cl R' = H, alkyl, aralkyl, thienyl, pyridyl, cycloalkyl or X-substd. mononuclear aryl A = alkylene, pref. ethylene or propylene B = a basic N-contng. radical with less than 12 C atoms, e.g. NH2, NHAlk, NAlk2 (preferred), piperidino, piperidyl, pyrrolidino, pyrrolidyl, morpholino, thiomorpholino, piperazino, homopiperazino, homopiperidino; all opt. substd. with 1 or more alkyl groups. n = 0 to 5 CNS depressants. |
