发明名称 BIOLOGICAL PREPARATION OF 13BETA-13-DEOXY-22,23- DIHYDROABELMEKUTIN-B1A/B1B AGLYCON
摘要 The known compound, 13 beta -13-deoxy-22,23-dihydro-avermectin -Bla/Blb Aglycone is prepared microbiologically from cultures of the novel microorganisms (MA-6762, ATCC 55069, MA-6763 ATCC 55070) or the known microorganism Streptomyces lavendulae MA-6555 (ATCC 14159). The compound is prepared by the biotransformation of 13-deoxy-22,23-dihydro avermectin Bla/Blb aglycone which oxidizes the 13-position and epimerizes the 13-position hydroxy group.
申请公布号 JPH04261180(A) 申请公布日期 1992.09.17
申请号 JP19910239615 申请日期 1991.09.19
申请人 MERCK & CO INC 发明人 KARINKA SHIYUMANOBU;REIMONDO EFU HOWAITO
分类号 A61K31/365;A61P33/10;C07D493/22;C12N1/20;C12P17/08;C12P17/18;C12R1/545;C12R1/56 主分类号 A61K31/365
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