发明名称 HYDROXYETHYLAMINO SULFONAMIDES USEFUL AS RETROVIRAL PROTEASE INHIBITORS
摘要 2140929 9404492 PCTABS00030 Hydroxyethylamino sulfonamide compounds of formulae (I, II) wherein R, R', R1, R1', R1'', R2, R3, R4, R6, x, t, Y, P1 and P2 are as defined in Claims 1 and 171, are effective as retroviral protease inhibitors, and in particular as inhibitors of HIV protease.
申请公布号 CA2140929(A1) 申请公布日期 1994.02.26
申请号 CA19932140929 申请日期 1993.08.24
申请人 SEARLE & CO;MONSANTO CO 发明人 VAZQUEZ MICHAEL L;MUELLER RICHARD A;TALLEY JOHN J;GETMAN DANIEL;DECRESCENZO GARY A;FRESKOS JOHN N
分类号 C07D295/12;A61K31/44;A61K31/4402;A61K31/4406;A61K31/4409;A61K31/4418;A61K31/4433;A61K31/505;A61K31/535;A61K31/5375;A61K38/00;A61P31/12;C07C311/05;C07C311/11;C07C311/13;C07C311/14;C07C311/18;C07C311/20;C07C311/24;C07C311/29;C07C311/32;C07C311/41;C07C311/46;C07C313/06;C07C317/04;C07C317/10;C07C317/14;C07C317/28;C07C317/44;C07C323/49;C07C323/57;C07C323/67;C07C327/38;C07D209/08;C07D211/78;C07D213/30;C07D213/53;C07D213/56;C07D213/64;C07D213/73;C07D213/81;C07D213/82;C07D213/89;C07D215/48;C07D233/54;C07D239/02;C07D239/26;C07D277/24;C07D277/30;C07D277/82;C07D307/20;C07D307/42;C07D307/79;C07D317/62;C07D333/34;C07D405/12;C07D409/12;C07D417/12;C07K5/06;C07K5/078;(IPC1-7):C07K5/06;C07D235/04;A61K38/05;C07D295/15;C07C311/19;A61K31/27;A61K31/33;C07D307/85 主分类号 C07D295/12
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