发明名称 |
NOVEL VITAMIN D ANALOGUES, THEIR PRODUCTION, USE THEREOF AND MEDICAMENTS CONTAINING THE SAME |
摘要 |
Vitamin D analogues of formula (I) are new. X = H or OH; R1, R2 = H or 1-3C alkyl; or CR1R2 = 3-6C carbocyclic ring; R3 = 1-3C alkyl, aryl, aralkyl or YR4; Y = C(O)S, C(S)O or C(S)S; R4 = 1-3C alkyl, aryl or aralkyl; Q = (CH2)n; R1, R2 and Q are all optionally substituted by one or more fluoro; and n = 1 to 4. |
申请公布号 |
HU9902689(A2) |
申请公布日期 |
1999.12.28 |
申请号 |
HU19990002689 |
申请日期 |
1997.05.15 |
申请人 |
LEO Pharmaceutical Products Ltd. A/S (Lovens Kemiske Fabrik Produktionsaktieselskab) |
发明人 |
BRETTING, CLAUS AAGE SVENSGAARD |
分类号 |
A61K31/59;C07C401/00 |
主分类号 |
A61K31/59 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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