发明名称 |
PROCESS FOR THE PREPARATION OF 2-AMINO-9-((2-PHENYL-1,3-DIOXAN-5-YLOXY)METHYL)-1H-PURIN-6(9H)-ONE COMPOUND USEFUL IN THE PREPARATION OF VALGANCICLOVIR |
摘要 |
The present invention provides an improved industrially feasible process for the preparation of 2-amino-9-((2-phenyl-1,3-dioxan-5-yloxy)methyl)-1H-purin-6(9H)-one, Formula which is a useful intermediate for the preparation of Valganciclovir and pharmaceutically acceptable salts thereof, and involves the use of said new intermediate compounds in the process to obtain Valganciclovir. |
申请公布号 |
EP2714691(B1) |
申请公布日期 |
2016.09.07 |
申请号 |
EP20110727115 |
申请日期 |
2011.05.31 |
申请人 |
PHARMATHEN S.A. |
发明人 |
KOFTIS, THEOCHARIS, V.;GEORGOPOULOU, IOANNA;VARVOGLI, ANASTASIA, AIKATERINI;ZITROU, ASTERIA |
分类号 |
C07D473/18 |
主分类号 |
C07D473/18 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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