发明名称 PROCESS FOR THE PREPARATION OF 2-AMINO-9-((2-PHENYL-1,3-DIOXAN-5-YLOXY)METHYL)-1H-PURIN-6(9H)-ONE COMPOUND USEFUL IN THE PREPARATION OF VALGANCICLOVIR
摘要 The present invention provides an improved industrially feasible process for the preparation of 2-amino-9-((2-phenyl-1,3-dioxan-5-yloxy)methyl)-1H-purin-6(9H)-one, Formula which is a useful intermediate for the preparation of Valganciclovir and pharmaceutically acceptable salts thereof, and involves the use of said new intermediate compounds in the process to obtain Valganciclovir.
申请公布号 EP2714691(B1) 申请公布日期 2016.09.07
申请号 EP20110727115 申请日期 2011.05.31
申请人 PHARMATHEN S.A. 发明人 KOFTIS, THEOCHARIS, V.;GEORGOPOULOU, IOANNA;VARVOGLI, ANASTASIA, AIKATERINI;ZITROU, ASTERIA
分类号 C07D473/18 主分类号 C07D473/18
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