发明名称 composto, formulação farmacêutica, uso de um composto, e, métodos para a inibição da atividade de bace e para o tratamento ou a prevenção de uma patologia relacionada a abeta em um mamífero
摘要 This invention relates to novel compounds having the structural formula I below: and to their pharmaceutically acceptable salt, compositions and methods of use. These novel compounds provide a treatment or prophylaxis of cognitive impairment, Alzheimer Disease, neurodegeneration and dementia.
申请公布号 BRPI0618845(A2) 申请公布日期 2016.09.13
申请号 BR2006PI18845 申请日期 2006.11.20
申请人 ASTEX THERAPEUTICS LIMITED;ASTRAZENECA AB 发明人 CHRISTOPHER MURRAY;GIANNI CHESSARI;JACOB KIHLSTRÖM;JEREMY BURROWS;JOHAN HEDSTRÖM;JOHAN LINDSTRÖM;KARIN KOLMODIN;KATARINA HÖGDIN;MILES STUART CONGREVE;SAHIL PATEL;STEFAN BERG;SVEN HELLBERG
分类号 C07D233/86;A61K31/4168;A61K31/4174;A61K31/4178;A61K31/427;A61K31/4439;A61K31/4725;A61K31/497;A61K31/506;A61K31/538;A61P25/16;A61P25/28;C07D233/88;C07D401/04;C07D401/10;C07D403/10;C07D405/04;C07D405/10;C07D405/14;C07D409/10;C07D413/10;C07D417/04 主分类号 C07D233/86
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