发明名称 |
composto, formulação farmacêutica, uso de um composto, e, métodos para a inibição da atividade de bace e para o tratamento ou a prevenção de uma patologia relacionada a abeta em um mamífero |
摘要 |
This invention relates to novel compounds having the structural formula I below: and to their pharmaceutically acceptable salt, compositions and methods of use. These novel compounds provide a treatment or prophylaxis of cognitive impairment, Alzheimer Disease, neurodegeneration and dementia. |
申请公布号 |
BRPI0618845(A2) |
申请公布日期 |
2016.09.13 |
申请号 |
BR2006PI18845 |
申请日期 |
2006.11.20 |
申请人 |
ASTEX THERAPEUTICS LIMITED;ASTRAZENECA AB |
发明人 |
CHRISTOPHER MURRAY;GIANNI CHESSARI;JACOB KIHLSTRÖM;JEREMY BURROWS;JOHAN HEDSTRÖM;JOHAN LINDSTRÖM;KARIN KOLMODIN;KATARINA HÖGDIN;MILES STUART CONGREVE;SAHIL PATEL;STEFAN BERG;SVEN HELLBERG |
分类号 |
C07D233/86;A61K31/4168;A61K31/4174;A61K31/4178;A61K31/427;A61K31/4439;A61K31/4725;A61K31/497;A61K31/506;A61K31/538;A61P25/16;A61P25/28;C07D233/88;C07D401/04;C07D401/10;C07D403/10;C07D405/04;C07D405/10;C07D405/14;C07D409/10;C07D413/10;C07D417/04 |
主分类号 |
C07D233/86 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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