发明名称 |
Crystalline salts of asenapine |
摘要 |
Disclosed is asenapine phosphate of formula (I) and its enantiomer (I) which can be used to prepare asenapine maleate. Further disclosed is a monoclinic crystalline form of asenapine maleate.; |
申请公布号 |
US9447109(B2) |
申请公布日期 |
2016.09.20 |
申请号 |
US201214113091 |
申请日期 |
2012.04.30 |
申请人 |
OLON S.P.A. |
发明人 |
Frigoli Samuele;Longoni Davide;Danelli Tamara;Alpegiani Marco |
分类号 |
C07D491/044 |
主分类号 |
C07D491/044 |
代理机构 |
Silvia Salvadori, PC. |
代理人 |
Silvia Salvadori, PC. ;Salvadori Silvia |
主权项 |
1. Asenapine phosphate of formula (I), or its enantiomer |
地址 |
Rodano IT |