发明名称 Pyrazolo(1,5-c)pyrimidine derivs - with hypnotic and tranquillizing activity
摘要 <p>Title derivs of formula (I): (where R1 and R4 are H, alkyl or aryl opt. mono- or disubst. by halogen, NO2, alkyl, alkoxy or alkylmercapto, R2 and R3 are H, halogen, NO2 or rhodanide, or R2 + R3 is alkylene, R5 is H, opt substd. alkyl or aryl opt. mono-or disubst. by NO2, halogen, alkyl, alkoxy, alkylmercapto, alkylamino or carboxyalkyl, and R6 and R7 are H, opt. subst. alkyl, alkenyl, cycloalkyl, alkoxyalkyl, or aryl opt. mono-or disubst. by halogen, lower alkyl, alkoxy, alkylmercapto, alkylamino or carboxyalkyl, or R6 + R7 is alkylene or alkenylene opt. substd. by lower alkyl and/or contg. O, S or N as a chain member, or R5 + R6 is alkylene and R7 has the above significance or is aryl, mono- or disubst. by halogen, NO2, lower alkyl, alkoxy, alkylmercapto or carboxyalkyl) may be prepd. by reacting a cpd. of formula R6R7N-CO-R5 with (I, -N=C(R5)-NR6R7 is NH2) in the presence of an inert solvent.</p>
申请公布号 DE2131790(A1) 申请公布日期 1973.01.11
申请号 DE19712131790 申请日期 1971.06.26
申请人 BAYER AG 发明人 KRANZ,ECKART,DR.;HOFFMEISTER,FRIEDRICH,DR.;WUTTKE,WOLFGANG,DR.
分类号 C07D487/04;(IPC1-7):C07D57/16 主分类号 C07D487/04
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