| 发明名称 |
Process for making hiv protease inhibitors |
| 摘要 |
<CHEM> Intermediates of structural formula (A) can be made by reacting a primary or secondary amine with glycidol or an activated derivative thereof. The process and intermediates are useful for synthesizing HIV protease inhibitor compounds, particularly L-735,524. <CHEM> |
| 申请公布号 |
AU7326794(A) |
申请公布日期 |
1995.02.13 |
| 申请号 |
AU19940073267 |
申请日期 |
1994.07.11 |
| 申请人 |
MERCK & CO., INC. |
发明人 |
DAVID ASKIN;PAUL REIDER;KAI ROSSEN;RICHARD J. VARSOLONA;KENNETH M WELLS |
| 分类号 |
A61K31/42;A61K31/423;A61K31/44;A61K31/495;A61K31/496;A61P31/12;A61P37/04;A61P43/00;C07D241/04;C07D263/52;C07D303/36;C07D401/06;C07D405/06;C07D413/06 |
主分类号 |
A61K31/42 |
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