发明名称 ONE POT SYNTHESIS OF 2-OXAZOLIDINONE DERIVATIVES
摘要 PROBLEM TO BE SOLVED: To provide a new process for preparing a compound of formula (I), by which the final product can be produced in a pure form in a high yield and in a large scale by the use of one pot procedure with respect to known processes, while avoiding the consumption of time and the necessity of high cost intermediate separation and further avoiding the necessity of dangerous reagents such as phosgene and environmentally injurious reagents such as tin chloride. SOLUTION: This one pot synthesis process for preparing (S)-4-ä[3-[2-(dimethylamino)ethyl]-1H-indol-5-yl]-methyl}-2-oxazolidinone. COPYRIGHT: (C)2006,JPO&NCIPI
申请公布号 JP2006225406(A) 申请公布日期 2006.08.31
申请号 JP20060152810 申请日期 2006.05.31
申请人 ASTRAZENECA AB 发明人 PATEL RAJNIKANT
分类号 C07D413/06;A61K31/00;A61K31/42;A61K31/421;A61K31/422;A61P25/00;A61P25/06;A61P43/00;C07B61/00;C07C215/06;C07C219/06;C07C219/32;C07C269/04;C07C269/06;C07C271/16;C07C271/20;C07C271/22;C07D209/14;C07D263/20 主分类号 C07D413/06
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