发明名称 |
PHARMACEUTICAL COMPOSITIONS CONTAINING 1-METHYL-3,6,7,8-TETRAHYDROPIRAZOLO[3,4-b]PIRROLO[4,3-d]PYRIDINE-6,8-DIONE DERIVATIVES, USE, AND PROCESS FOR PREPARING THEM |
摘要 |
<p>The present invention is related to new derivatives of 1-methyl-3,6,7,8- tetrahydropirazolo[3,4-b]pirrolo[4,3-d]piridin-6,8-dione nucleus, preferably heterocyclic derivatives, acting as hypnotics and analgesic in the central nervous system, being useful in the treatment of anxiety and central hyperalgesia, including: anxiety relief, central hyperalgesia relief in mammals, preferably humans. It is also described pharmaceutical compositions containing said compounds and preparation processes.</p> |
申请公布号 |
WO2006092032(A2) |
申请公布日期 |
2006.09.08 |
申请号 |
WO2006BR00037 |
申请日期 |
2006.03.03 |
申请人 |
UNIVERSIDADE FEDERAL DO RIO DE JANEIRO - UFRJ;DE LACERDA BARREIRO, ELIEZER DE JESUS;MANSSOUR FRAGA, CARLOS ALBERTO;ZAPATA SUDO, GISELE;TAKASHI SUDO, ROBERTO;MENEGATTI, RICARDO |
发明人 |
DE LACERDA BARREIRO, ELIEZER DE JESUS;MANSSOUR FRAGA, CARLOS ALBERTO;ZAPATA SUDO, GISELE;TAKASHI SUDO, ROBERTO;MENEGATTI, RICARDO |
分类号 |
C07D471/12;C07D471/14;A61K31/437;A61P25/00;A61P25/04;A61P25/28 |
主分类号 |
C07D471/12 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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