发明名称 PHARMACEUTICAL COMPOSITIONS CONTAINING 1-METHYL-3,6,7,8-TETRAHYDROPIRAZOLO[3,4-b]PIRROLO[4,3-d]PYRIDINE-6,8-DIONE DERIVATIVES, USE, AND PROCESS FOR PREPARING THEM
摘要 <p>The present invention is related to new derivatives of 1-methyl-3,6,7,8- tetrahydropirazolo[3,4-b]pirrolo[4,3-d]piridin-6,8-dione nucleus, preferably heterocyclic derivatives, acting as hypnotics and analgesic in the central nervous system, being useful in the treatment of anxiety and central hyperalgesia, including: anxiety relief, central hyperalgesia relief in mammals, preferably humans. It is also described pharmaceutical compositions containing said compounds and preparation processes.</p>
申请公布号 WO2006092032(A2) 申请公布日期 2006.09.08
申请号 WO2006BR00037 申请日期 2006.03.03
申请人 UNIVERSIDADE FEDERAL DO RIO DE JANEIRO - UFRJ;DE LACERDA BARREIRO, ELIEZER DE JESUS;MANSSOUR FRAGA, CARLOS ALBERTO;ZAPATA SUDO, GISELE;TAKASHI SUDO, ROBERTO;MENEGATTI, RICARDO 发明人 DE LACERDA BARREIRO, ELIEZER DE JESUS;MANSSOUR FRAGA, CARLOS ALBERTO;ZAPATA SUDO, GISELE;TAKASHI SUDO, ROBERTO;MENEGATTI, RICARDO
分类号 C07D471/12;C07D471/14;A61K31/437;A61P25/00;A61P25/04;A61P25/28 主分类号 C07D471/12
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