发明名称 NEW TRIAZOLOPURINES, METHOD OF PREPARING THEM AND THEIR USE AS DRUGS
摘要 The invention pertains to triazolopurines of formula (I). The claimed compounds show an affinity to adenosine receptors and thus represent a new class of adenosine antagonists. Generally, adenosine antagonists can have a therapeutically useful effect in cases where diseases or pathological situations involve activation of adenosine receptors.
申请公布号 CA2256736(A1) 申请公布日期 1998.01.29
申请号 CA19972256736 申请日期 1997.07.17
申请人 BOEHRINGER INGELHEIM INTERNATIONAL GMBH 发明人 GAIDA, WOLFRAM;WEISER, THOMAS;POHL, GERALD;MIERAU, JOACHIM;LEHR, ERICH;KUEFNER-MUEHL, ULRIKE;KUMMER, WERNER
分类号 A61K31/00;A61K31/505;A61K31/519;A61K31/529;A61K31/535;A61K31/5375;A61K31/5377;A61P5/36;A61P7/00;A61P7/10;A61P11/00;A61P11/06;A61P13/00;A61P13/12;A61P19/00;A61P19/02;A61P25/06;A61P25/16;A61P25/24;A61P25/28;A61P37/00;A61P43/00;C07D235/00;C07D239/00;C07D249/00;C07D487/14;(IPC1-7):C07D473/18;A61K31/52;A61K31/53;A61K31/54 主分类号 A61K31/00
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