发明名称 |
Process for preparing Estrogen-antagonistic 11 beta-Fluoro-17alpha-alkylestra-1,3,5(10)-triene-3,17-diols having a 7alpha-(xi-Alkylamino-omega-perfluoroalkyl)alkyl side chain and alpha-Alkyl(amino)-omega-perfluoro(alkyl)alkanes and Processes for their Preparation |
摘要 |
The present invention relates to a new process for preparing estrogen-antagonistic 11beta-fluoro-17alpha-alkylestra-1,3,5(10)-triene-3,17-diols of the general formula I having a 7alpha-(xi-alkylamino-omega-perfluoroalkyl)alkyl side chain and to alpha-alkyl(amino)-omega-perfluoro(alkyl)alkanes of the general formula II, to processes for their preparation and to the intermediates required for this purpose.
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申请公布号 |
US2009062558(A1) |
申请公布日期 |
2009.03.05 |
申请号 |
US20080201043 |
申请日期 |
2008.08.29 |
申请人 |
SANDER MICHAEL;GROSSBACH DANJA;DINTER CHRISTIAN;HASSFELD JORMA;VOIGTLAENDER DAVID |
发明人 |
SANDER MICHAEL;GROSSBACH DANJA;DINTER CHRISTIAN;HASSFELD JORMA;VOIGTLAENDER DAVID |
分类号 |
C07J1/00;C07C19/08;C07C211/00;C07F9/02 |
主分类号 |
C07J1/00 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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