发明名称 Process for preparing Estrogen-antagonistic 11 beta-Fluoro-17alpha-alkylestra-1,3,5(10)-triene-3,17-diols having a 7alpha-(xi-Alkylamino-omega-perfluoroalkyl)alkyl side chain and alpha-Alkyl(amino)-omega-perfluoro(alkyl)alkanes and Processes for their Preparation
摘要 The present invention relates to a new process for preparing estrogen-antagonistic 11beta-fluoro-17alpha-alkylestra-1,3,5(10)-triene-3,17-diols of the general formula I having a 7alpha-(xi-alkylamino-omega-perfluoroalkyl)alkyl side chain and to alpha-alkyl(amino)-omega-perfluoro(alkyl)alkanes of the general formula II, to processes for their preparation and to the intermediates required for this purpose.
申请公布号 US2009062558(A1) 申请公布日期 2009.03.05
申请号 US20080201043 申请日期 2008.08.29
申请人 SANDER MICHAEL;GROSSBACH DANJA;DINTER CHRISTIAN;HASSFELD JORMA;VOIGTLAENDER DAVID 发明人 SANDER MICHAEL;GROSSBACH DANJA;DINTER CHRISTIAN;HASSFELD JORMA;VOIGTLAENDER DAVID
分类号 C07J1/00;C07C19/08;C07C211/00;C07F9/02 主分类号 C07J1/00
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