发明名称 USE OF BICYCLIC ESTERS OR AMIDES FOR THE TREATMENT OF DISEASES RESPONSIVE TO ENHANCED POTASSIUM CHANNEL ACTIVITY
摘要 A compound of formula (I): or a salt, solvate or physiologically functional derivative thereof for use as a IK and/or SK channel opener. Methods of screening SK ion channels, particularly SK1 and medicaments for the treatment of a urinogenital, respiratory, cardiovascular, neuronal disorder, of sleeping disorders, sickle cell anemia, pain, inflammation and bowel disease (IBD) are also disclosed.
申请公布号 WO02062745(A1) 申请公布日期 2002.08.15
申请号 WO2002GB00496 申请日期 2002.02.04
申请人 GLAXO GROUP LIMITED;COX, BRIAN;CRYAN, JENNIFER, ELIZABETH;DALE, TIMOTHY, JAMES;ROBERTSON, GRAEME, MICHAEL;TREZISE, DEREK, JOHN 发明人 COX, BRIAN;CRYAN, JENNIFER, ELIZABETH;DALE, TIMOTHY, JAMES;ROBERTSON, GRAEME, MICHAEL;TREZISE, DEREK, JOHN
分类号 G01N33/50;A61K31/165;A61K31/35;A61K31/38;A61K31/44;A61K31/535;A61K45/00;A61P1/04;A61P7/06;A61P9/00;A61P9/10;A61P9/12;A61P11/00;A61P11/06;A61P13/00;A61P15/00;A61P25/00;A61P25/02;A61P25/18;A61P25/20;A61P29/00;C07C233/11;C07C235/34;C07D215/12;C07D295/185;C07D311/58;C07D335/06;G01N33/15;(IPC1-7):C07C233/11;C07D295/18;C07D223/16 主分类号 G01N33/50
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