发明名称 |
CARBAMATE-SUBSTITUTED OXINDOLE DERIVATIVES AND USE THEREOF FOR THE TREATMENT OF VASOPRESSIN-DEPENDENT DISEASES |
摘要 |
The invention relates to novel carbamate-substituted oxindole derivatives of formula (I), pharmaceuticals containing the same, and the use thereof for treating vasopressin-dependent diseases. In said formula (I), R1 represents hydrogen, methoxy, or ethoxy, R2 represents hydrogen or methoxy, R3 represents hydrogen, methyl, ethyl, n-propyl, or isopropyl, and X1 and X2 represent N or CH, provided that X1 and X2 do not simultaneously represent N. |
申请公布号 |
WO2010009775(A1) |
申请公布日期 |
2010.01.28 |
申请号 |
WO2008EP66933 |
申请日期 |
2008.12.05 |
申请人 |
ABBOTT GMBH & CO. KG;NETZ, ASTRID;OOST, THORSTEN;GENESTE, HERVE;BRAJE, WILFRIED;WERNET, WOLFGANG;UNGER, LILIANE;HORNBERGER, WILFRIED;LUBISCH, WILFRIED |
发明人 |
NETZ, ASTRID;OOST, THORSTEN;GENESTE, HERVE;BRAJE, WILFRIED;WERNET, WOLFGANG;UNGER, LILIANE;HORNBERGER, WILFRIED;LUBISCH, WILFRIED |
分类号 |
C07D401/14;A61K31/4545;A61K31/496;A61P3/10;A61P7/02 |
主分类号 |
C07D401/14 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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