| 发明名称 |
A PREPARATION METHOD OF CANDESARTAN CILEXETIL AND INTERMEDIATES THEREOF |
| 摘要 |
A preparation method of candesartan cilexetil and intermediates thereof. A compound of formula I, wherein R1 is chloride, bromide, iodide, hydroxy, sulfonyl, mesyl, p-tosyloxy, methanesulfonyloxy, acetoxy, benzoyloxy, or dimethylmercapto group. A preparation method of candesartan cilexetil from the compound of formula I. The material used in the method is stable. |
| 申请公布号 |
WO2009003339(A1) |
申请公布日期 |
2009.01.08 |
| 申请号 |
WO2007CN70214 |
申请日期 |
2007.06.29 |
| 申请人 |
TOPHARMAN SHANGHAI CO., LTD.;SHANGHAI INSTITUTE OF MATERIA MEDICA, CHINESE ACADEMY OF SCIENCES;LI, HAIHONG;JIANG, XIANGRUI;ZHAO, QINGJIE;YANG, CHI;SHEN, JINGSHAN |
发明人 |
LI, HAIHONG;JIANG, XIANGRUI;ZHAO, QINGJIE;YANG, CHI;SHEN, JINGSHAN |
| 分类号 |
C07D403/10 |
主分类号 |
C07D403/10 |
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