发明名称 PROCESS FOR THE PREPARATION OF PYRIMIDINE COMPOUNDS
摘要 <p>A process for preparing a compound of formula (I) comprising treating a compound of formula (II) with either (a) an acid catalyst optionally in the presence of a means for removing methanol, or (b) an acid chloride; provided that when the acid catalyst is <u>p</u>-toluene sulphonic acid or potassium bisulphite then the process is conducted in the presence of an acid anhydride.</p>
申请公布号 WO9807707(A1) 申请公布日期 1998.02.26
申请号 WO1997GB02015 申请日期 1997.07.25
申请人 ZENECA LIMITED;BERRY, IAN, GORDON;COX, BRIAN, JEFFREY;DE BOOS, GARETH, ANDREW;FLEMING, IAN, GEORGE;JONES, RAYMOND, VINCENT, HEAVON;WHITTON, ALAN, JOHN 发明人 BERRY, IAN, GORDON;COX, BRIAN, JEFFREY;DE BOOS, GARETH, ANDREW;FLEMING, IAN, GEORGE;JONES, RAYMOND, VINCENT, HEAVON;WHITTON, ALAN, JOHN
分类号 C07D239/34;(IPC1-7):C07D239/34 主分类号 C07D239/34
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