发明名称 |
2,3,4,5-TETRAHYDRO-1H-[1,4]BENZODIAZEPINE-3-HYDROXAMIC ACID AS MATRIX METALLOPROTEINASE INHIBITORS |
摘要 |
Compounds having formula (1) are useful in treating disease conditions mediated by matrix metalloproteinases and TACE, such as tumor growth, osteoarthritis, rheumatoid arthritis and degenerative cartilage loss.
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申请公布号 |
WO0044730(A1) |
申请公布日期 |
2000.08.03 |
申请号 |
WO2000US01991 |
申请日期 |
2000.01.27 |
申请人 |
AMERICAN CYANAMID COMPANY |
发明人 |
ALBRIGHT, JAY, DONALD;DELOS SANTOS, EFREN, GUILLERMO;LEVIN, JEREMY, IAN;CHEN, JAMES, MING |
分类号 |
C07D243/16;A61K31/5513;A61P1/02;A61P1/14;A61P1/16;A61P3/10;A61P9/10;A61P13/12;A61P15/00;A61P17/00;A61P19/02;A61P19/04;A61P19/08;A61P25/28;A61P27/02;A61P29/00;A61P31/04;A61P31/18;A61P35/00;A61P37/06;A61P43/00;C07D243/14;C07D401/06;C07D403/10;C07D405/06;C07D409/06;(IPC1-7):C07D243/14;C07D521/00;A61K31/551 |
主分类号 |
C07D243/16 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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