发明名称 AMINOQUINAZOLINE COMPOUNDS AS A2A ANTAGONIST
摘要 The present invention is directed to compounds of generic formula I: or pharmaceutically acceptable salts thereof that are believed to be useful as an A2A-receptor antagonist.
申请公布号 WO2016126570(A1) 申请公布日期 2016.08.11
申请号 WO2016US15881 申请日期 2016.02.01
申请人 MERCK SHARP & DOHME CORP.;ALI, AMJAD;ZHOU, GANG;KUANG, RONGZE;LIM, YEON-HEE;LO, MICHAEL MAN-CHU;TING, PAULINE, C.;BIJU, PURAKKATTLE;RUIZ, MANUEL DE LERA;DEGRADO, SYLVIA, J.;TUNG, ALEXANDER, L.;HENDERSON, TIMOTHY, J.;HONG, LIWU;KIM, JAE-HUN;KIM, DAVID WON-SHIK;LEE, JOE, F.;WU, JIE;WU, HEPING;XIAO, YUSHI;YU, TAO;ZHU, XIAOHONG;MCCORMICK, KEVIN, D.;TAGAT, JAYARAM, R.;XIAO, DONG;KHAN, TANWEER;CAO, JIANHUA;BERLIN, MICHAEL;ZHANG, YONGLIAN 发明人 ALI, AMJAD;ZHOU, GANG;KUANG, RONGZE;LIM, YEON-HEE;LO, MICHAEL MAN-CHU;TING, PAULINE, C.;BIJU, PURAKKATTLE;RUIZ, MANUEL DE LERA;DEGRADO, SYLVIA, J.;TUNG, ALEXANDER, L.;HENDERSON, TIMOTHY, J.;HONG, LIWU;KIM, JAE-HUN;KIM, DAVID WON-SHIK;LEE, JOE, F.;WU, JIE;WU, HEPING;XIAO, YUSHI;YU, TAO;ZHU, XIAOHONG;MCCORMICK, KEVIN, D.;TAGAT, JAYARAM, R.;XIAO, DONG;KHAN, TANWEER;CAO, JIANHUA;BERLIN, MICHAEL;ZHANG, YONGLIAN
分类号 A61K31/517;C07D239/84;C07D403/12 主分类号 A61K31/517
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