发明名称 5-(2-imidazolinylamino)-benzimidazole derivatives, their preparation and their use as .alpha.-adrenoceptor agonists with improved metabolic stability
摘要 Benzimidazole compounds having the generic structure:are used to treat alpha-2 mediated disorders, including nasal congestion, glaucoma, asthma, migraine, and diarrhea.
申请公布号 US6486190(B1) 申请公布日期 2002.11.26
申请号 US20000554698 申请日期 2000.05.18
申请人 THE PROCTER & GAMBLE COMPANY 发明人 CUPPS THOMAS LEE;BOGDAN SOPHIE EVA;NIKOLAIDES NICK;GILBERT SHERI ANN;GAZDA MICHAEL;DOBSON ROY LEE;CRUZE CHARLES ANDREW III
分类号 A61K31/4184;A61P1/00;A61P11/00;A61P25/00;A61P25/04;A61P25/06;A61P27/02;A61P27/06;A61P29/00;A61P31/12;A61P37/08;A61P43/00;C07D403/12;(IPC1-7):A61K31/418 主分类号 A61K31/4184
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