发明名称 |
FORMATION OF N-PROTECTED BIS-3,6-(4-AMINOBUTYL)-2,5-DIKETOPIPERAZ INE THROUGH A CYCLIC ALPHA-N-PROTECTED AMINO ESTER. |
摘要 |
A method for the synthesis of N-protected 3,6-aminoalkyl-2,5-diketopiperazines is provided. The method includes obtaining a cyclic a-N protected active amino ester and adding it to a mixture of an amine catalyst in an organic solvent. |
申请公布号 |
MX2015012603(A) |
申请公布日期 |
2016.06.10 |
申请号 |
MX20150012603 |
申请日期 |
2014.03.14 |
申请人 |
MANNKIND CORP. |
发明人 |
JOHN J. FREEMAN;OTTO PHANSTIEL;WILLIAMS ELLIOT BAY;KELLY SULLIVAN KRAFT |
分类号 |
C07D241/10 |
主分类号 |
C07D241/10 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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