发明名称 BENZOHETEROCYCLIC COMPOUNDS
摘要 Novel benzoheterocyclic compound of formula (I) and pharmaceutically acceptable salts thereof, which show excellent antivasopressin activity and oxytocin antagonistic activity, and are useful as a vasopressin antagonist or oxytocin antagonist. A is a 5- or 6-membered unsaturated heterocyclic residue having 1 to 2 heteroatoms. B1 and B2 are each methylene or a group of the formula: -NR8- (wherein R8 is a hydrogen atom or a lower alkyl group).
申请公布号 CA2120916(A1) 申请公布日期 1994.03.03
申请号 CA19932120916 申请日期 1993.08.03
申请人 OTSUKA PHARMA CO LTD 发明人 OGAWA HIDENORI;KONDO KAZUMI;YAMASHITA HIROSHI;KAN KEIZO;TOMINAGA MICHIAKI;YABUUCHI YOICHI
分类号 C22F1/00;A61K31/55;C07D401/06;C07D401/14;C07D405/06;C07D405/14;C07D409/06;C07D409/14;C07D413/14;C07D417/06;C07D417/14;H01B12/10;(IPC1-7):C07D401/06 主分类号 C22F1/00
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