发明名称 QUINOLINE DERIVATIVE
摘要 This compound represented by general formula (I) and having a quinoline skeleton has a strong Axl inhibitory activity. Consequently, this compound can be a therapeutic agent for Axl-related diseases, for example, cancers such as acute myeloid leukemia, chronic myeloid leukemia, melanoma, breast cancer, pancreatic cancer and glioma, kidney diseases, immune system diseases and cardiovascular diseases.
申请公布号 WO2016104617(A1) 申请公布日期 2016.06.30
申请号 WO2015JP86050 申请日期 2015.12.24
申请人 ONO PHARMACEUTICAL CO., LTD. 发明人 INUKAI, TAKAYUKI;TAKEUCHI, JUN;YASUHIRO, TOMOKO
分类号 C07D401/14;A61K31/4709;A61K31/517;A61K31/55;A61P7/02;A61P9/00;A61P9/10;A61P13/12;A61P17/06;A61P19/02;A61P29/00;A61P35/00;A61P35/02;A61P35/04;A61P43/00;C07D471/04 主分类号 C07D401/14
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