发明名称 Indanol derivative
摘要 The present invention provides a compound having the following general formula (I) which is useful as a neurokinin receptor antagonist: (wherein, R<SUP>1</SUP>, R<SUP>2</SUP>: optionally substituted (hetero)aryl, R<SUP>3</SUP>: -CO-R<SUP>4</SUP>, -CO-O-R<SUP>4</SUP>, etc., R<SUP>4</SUP>: alkyl, cycloalkyl, etc., A: CH<SUB>2</SUB>, CO, SO<SUB>2</SUB>, B: a single bond, etc., D: oxygen, CH<SUB>2</SUB>, E: alkylene, alkenylene, n: 1 to 3).
申请公布号 US7365067(B2) 申请公布日期 2008.04.29
申请号 US20050590305 申请日期 2005.02.24
申请人 SANKYO COMPANY, LIMITED 发明人 NISHI TAKAHIDE;TAKEMOTO TOSHIYASU;IKEDA TAKUYA;MORIMOTO KIYOSHI
分类号 A61K31/5377;A61P1/00;A61P1/04;A61P1/08;A61P1/12;A61P7/12;A61P9/00;A61P9/10;A61P11/00;A61P11/02;A61P11/06;A61P11/08;A61P11/14;A61P13/10;A61P17/00;A61P17/04;A61P17/06;A61P19/02;A61P19/04;A61P25/02;A61P25/04;A61P25/06;A61P25/18;A61P25/22;A61P25/24;A61P25/28;A61P25/30;A61P27/02;A61P29/00;A61P37/02;A61P37/08;A61P43/00;C07D413/06;C07D413/14 主分类号 A61K31/5377
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