发明名称 NEW PIPERIDINE, TETRAHYDROPYRIDINE AND PYRROLIDINE DERIVATIVES, PROCESS FOR PREPARING THESE AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
摘要 The invention relates to compounds of formula I: <IMAGE> in which R1 represents a naphthyl radical, a dihydronaphthyl radical, a tetrahydronaphthyl radical, a quinolyl radical or a 1,4-benzodioxanyl radical, A represents a single bond, a double bond, a methylene radical, a radical of formula z1: -CH=(z1) or a radical of formula z2: =CH-(z2) the ring B represents a piperidyl radical, a pyrrolidinyl radical, or a 1,2,3,6-tetrahydropyridyl radical, and R2 represents: a hydrogen atom, a benzyl radical, or an alkyl radical having 1 to 6 carbon atoms, on condition that in one of these cases R1 is other than a naphthyl (y1), dihydronaphthyl (y2) or tetrahydronaphthyl (y3) radical and B is other than a piperidinyl radical, or an aminoalkyl radical having 1 to 6 carbon atoms, a cyanoalkyl radical having 1 to 6 carbon atoms, or a radical of formula w1: <IMAGE> (w1) in which n is 1-6 and R4 represents a hydrogen atom, a halogen atom, an alkyl radical having 1 to 6 carbon atoms, or an alkoxy radical having 1 to 6 carbon atoms , and their addition salts with a pharmaceutically-acceptable inorganic or organic acid, and medicaments containing the same.
申请公布号 AU8025191(A) 申请公布日期 1992.01.16
申请号 AU19910080251 申请日期 1991.07.09
申请人 ADIR ET COMPAGNIE 发明人 GILBERT LAVIELLE;MICHEL LAUBIE;FRANCIS COLPAERT
分类号 A61K31/40;A61K31/4025;A61K31/44;A61K31/4427;A61K31/443;A61K31/445;A61K31/4465;A61K31/451;A61K31/47;A61P9/12;A61P25/04;A61P25/18;A61P25/20;A61P25/24;A61P25/26;A61P43/00;C07D207/06;C07D207/08;C07D207/20;C07D211/12;C07D211/14;C07D211/18;C07D211/22;C07D211/70;C07D295/13;C07D295/185;C07D401/04;C07D401/06;C07D405/04;C07D405/06 主分类号 A61K31/40
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