发明名称 AZETIDINONE DERIVATIVES AND METHODS OF USE THEREOF
摘要 <p>The present invention relates to methods for treating or preventing a disorder of lipid metabolism, pain, diabetes, a vascular condition, demyelination or nonalcoholic fatty liver disease, comprising administering a compound having the formula (I) or a pharmaceutically acceptable salt, solvate, ester, prodrug or stereoisomer thereof, wherein: R&lt;SUP&gt;1&lt;/SUP&gt; and R&lt;SUP&gt;2&lt;/SUP&gt; are defined in Tables 1-6 herein, and R&lt;SUB&gt;3&lt;/SUB&gt; is -phenyl, -4-chlorophenyl, -2-pyridyl, or -3-pyridyl.</p>
申请公布号 WO2008033465(A1) 申请公布日期 2008.03.20
申请号 WO2007US19931 申请日期 2007.09.13
申请人 SCHERING CORPORATION;ASLANIAN, ROBERT, G.;CHAN, TIN-YAU;HARRIS, JOEL, M.;MCKITTRICK, BRIAN, A.;NEUSTADT, BERNARD, R.;PALANI, ANANDAN;PRIESTLEY, TONY;SMITH, ELIZABETH, M.;STAMFORD, ANDREW, W.;VACCARO, HENRY, M.;XIAO, DONG 发明人 ASLANIAN, ROBERT, G.;CHAN, TIN-YAU;HARRIS, JOEL, M.;MCKITTRICK, BRIAN, A.;NEUSTADT, BERNARD, R.;PALANI, ANANDAN;PRIESTLEY, TONY;SMITH, ELIZABETH, M.;STAMFORD, ANDREW, W.;VACCARO, HENRY, M.;XIAO, DONG
分类号 A61K31/4427;A61P3/06;A61P3/10;A61P9/10;A61P25/28;C07D401/04 主分类号 A61K31/4427
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