发明名称 Pharmaceutical formulations, processes, solid forms and methods of use relating to 1-ethyl-7-(2-methyl-6-(1H-1,2,4-triazol-3-yl)pyridin-3-yl)-3,4-dihydropyrazino[2,3-b] pyrazin-2(1H)-one
摘要 Provided herein are formulations, processes, solid forms and methods of use relating to 1-ethyl-7-(2-methyl-6-(1H-1,2,4-triazol-3-yl)pyridin-3-yl)-3,4-dihydropyrazino[2,3-b]pyrazin-2(1H)-one.
申请公布号 US9359364(B2) 申请公布日期 2016.06.07
申请号 US201414254023 申请日期 2014.04.16
申请人 Signal Pharmaceuticals, LLC 发明人 Menon Anil;Parikh Darshan K.;Visky Dora;Kreilein Matthew Michael;Boersen Nathan;Lee Thomas;Li Ying;Xu Jean;Liang Xiaozhang;Leong William Wei-Hwa;Cohen Benjamin
分类号 C07D487/04;A61K31/4985;C07D471/04;A61K9/20;A61K9/48 主分类号 C07D487/04
代理机构 Jones Day 代理人 Jones Day
主权项 1. A crystal form of Compound 1, or a tautomer thereof:which has an X-ray powder diffraction pattern comprising peaks at 9.8±0.2, 12.0±0.2 and 17.9±0.2° 2θ.
地址 San Diego CA US