发明名称 |
Monomeric and dimeric nucleosides with silyl-containing diamino phosphorous linkages |
摘要 |
Synthetic processes are provided wherein substituted silylalkyl phosphoramidites serve as coupling reagents for preparing phosphate, phosphorothioate, and other phosphorous-containing covalent linkages. Also provided are synthetic intermediates useful in such processes. h processes.
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申请公布号 |
US5847106(A) |
申请公布日期 |
1998.12.08 |
申请号 |
US19970789443 |
申请日期 |
1997.01.27 |
申请人 |
ISIS PHARMACEUTICALS INC. |
发明人 |
RAVIKUMAR, VASULINGA;MULVEY, DENNIS;COLE, DOUGLAS L.;COOK, PHILLIP DAN |
分类号 |
C07H19/06;A61K31/70;A61K31/7042;A61K31/7052;A61K31/7064;A61K31/7068;A61K31/7072;A61K31/7076;A61K31/708;A61K31/7088;A61P31/12;A61P35/00;C07F9/146;C07F9/24;C07H19/16;C07H21/00;C07H21/02;C07H21/04;C07H23/00;(IPC1-7):C07H21/00 |
主分类号 |
C07H19/06 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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