发明名称 PROCESS FOR THE PREPARATION OF (R)-3-(4-(7H-PYRROLO[2,3-D], PYRIMIDIN-4-YL)-1 H-PYRAZOL-1-YL)-3-CYCLOPENTYLPROPANENITRILE PHOSPHATE AND ITS POLYMORPHS THEREOF
摘要 The present invention provides an improved process for the preparation of (R)-3-(4-(7H- pyrrolo[2,3d-]pyrimidin-4-yl)-lH-pyrazol-l-yl)-3-cyclopentylpropanenitrile phosphate compound of formula- la and its novel polymorphs thereof, which is represented by the following structural formula:
申请公布号 WO2016063294(A3) 申请公布日期 2016.07.07
申请号 WO2015IN00398 申请日期 2015.10.20
申请人 MSN LABORATORIES PRIVATE LIMITED;THIRUMALAI RAJAN, SRINIVASAN;ESWARAIAH, SAJJA;VENKATA PANAKALA RAI, GOGULAPATI 发明人 THIRUMALAI RAJAN, SRINIVASAN;ESWARAIAH, SAJJA;VENKATA PANAKALA RAI, GOGULAPATI
分类号 C07D487/04;A61K31/519 主分类号 C07D487/04
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