发明名称 SUBSTITUTED 1-AZOLYL-BUTAN-2-ONES,PROCESSES FOR THEIR PREPARATION AND THEIR USE AS FUNGICIDES AND AS INTERMEDIATE PRODUCTS
摘要 1. Substituted 1-azolyl-butan-2-ones of the formula see diagramm : EP0054865,P68,F1 in which Az represents 1,2,4-triazol-1-yl and 4-yl or imidazol-1-yl ; R**1 represents hydrogen, alkyl with 1 to 12 and alkenyl and alkinyl with in each case 2 to 12 carbon atoms, and represents optionally C1 -C4 -alkyl-substituted cycloalkyl with 3 to 7 carbon atoms or cycloalkylalkyl with 3 to 7 carbon atoms in the cycloalkyl part and 1 to 4 carbon atoms in the alkyl part, and represents optionally substituted phenoxyalkyl with 1 to 4 carbon atoms in the alkyl part or optionally substituted phenylalkyl with 1 to 4 carbon atoms in the alkyl part, the phenyl substituents to be mentioned in each case being : halogen ; alkyl, alkoxy and alkylthio with in each case 1 to 6 carbon atoms ; cyclohexyl ; dialkylamino with in each case 1 to 4 carbon atoms in each alkyl part ; halogenoalkyl, halogenoalkoxy and halogenoalkylthio with in each case 1 to 4 carbon atoms and 1 to 5 identical or different halogen atoms ; nitro ; cyano ; alkoxycarbonyl with 1 to 4 carbon atoms in the alkyl part ; and optionally halogensubstituted phenyl and phenoxy ; and the grouping -CO-NR**6 R**7 ; n represents the numbers 0 or 1, R**2 represents cyano or the groupings -X-R**3 and -CO-NR**4 R**5 , and, in the case where n does not represent 0 at the same time as R**1 represents hydrogen and Az represents 1,2,4-triazolyl, also additionally represents optionally substituted aryl with 6 to 10 carbon atoms, possible substituents being the aryl substituents already mentioned under R**1 , and represents alkoxycarbonyl with 1 to 4 carbon atoms in the alkyl part ; X represents oxygen, sulphur, or the SO or SO2 group, R**3 represents alkyl with 1 to 6 carbon atoms, halogenoalkyl with 1 to 4 carbon atoms and 1 to 5 identical or different halogen atoms, and represents optionally substituted aryl with 6 to 10 carbon atoms and aralkyl with 6 to 10 carbon atoms in the aryl part and 1 to 2 carbon atoms in the alkyl part, possible substituents being the aryl substituents already mentioned under R**1 ; R**4 represents hydrogen, alkyl with 1 to 4 carbon atoms or optionally substituted aryl with 1 to 10 carbon atoms, possible substituents being the aryl substituents already mentioned under R**1 ; R**5 represents hydrogen or alkyl with 1 to 4 carbon atoms ; and R**6 and R**7 represent hydrogen, alkyl with 1 to 4 carbon atoms, phenyl which is optionally substituted by halogen and alkyl with 1 to 4 carbon atoms, or both together with the adjacent nitrogen atom represent a saturated 5- or 6-membered ring system which can contain nitrogen or oxygen as additional hetero atoms ; and plant-tolerated acid addition salts and metal salt complexes thereof.
申请公布号 ZA8108757(B) 申请公布日期 1982.11.24
申请号 ZA19810008757 申请日期 1981.12.18
申请人 BAYER AG 发明人 KRAEMER W;BUECHEL K;ELBE H;KRAATZ U;REGEL E;FROHBERGER P;BRANDES W
分类号 A01N43/50;A01N43/64;A01N43/653;A01N47/02;C07C45/63;C07C45/67;C07C45/71;C07C49/16;C07D233/60;C07D249/08;C07D521/00 主分类号 A01N43/50
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