发明名称 COMPOUNDS AND METHODS FOR INHIBITING THE INTERACTION OF BCL PROTEINS WITH BINDING PARTNERS
摘要 The invention relates to isoxazolidine containing compounds that bind to bcl proteins and inhibit BcI function. The compounds may be used for treating and modulating disorders associated with hyperproliferation, such as cancer.
申请公布号 WO2008024337(A2) 申请公布日期 2008.02.28
申请号 WO2007US18471 申请日期 2007.08.21
申请人 INFINITY DISCOVERY, INC.;CASTRO, ALFREDO, C.;DEPEW, KRISTOPHER, M.;GROGAN, MICHAEL, J.;HOLSON, EDWARD, B.;HOPKINS, BRIAN, T.;JOHANNES, CHARLES, W.;KEANEY, GREGG, F.;KONEY, NII, O.;LIU, TAO;MANN, DAVID, A.;NEVALAINEN, MARTA;PELUSO, STEPHANE;PEREZ, LAWRENCE, BLAS;SNYDER, DANIEL, A.;TIBBITTS, THOMAS, T. 发明人 CASTRO, ALFREDO, C.;DEPEW, KRISTOPHER, M.;GROGAN, MICHAEL, J.;HOLSON, EDWARD, B.;HOPKINS, BRIAN, T.;JOHANNES, CHARLES, W.;KEANEY, GREGG, F.;KONEY, NII, O.;LIU, TAO;MANN, DAVID, A.;NEVALAINEN, MARTA;PELUSO, STEPHANE;PEREZ, LAWRENCE, BLAS;SNYDER, DANIEL, A.;TIBBITTS, THOMAS, T.
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