发明名称 Glikokinaz aktivatörleri
摘要 Mevcut bulus, formül (I)'in R1,R2,R3, ve R4'ün istem 1 'de tanimlandigi gibi oldugu bilesikleri ve bunlarin farmasötik açidan kabul edilebilir tuzlari ile ilgilidir. Bilesikler, tip II diyabetin tedavisinde ensülin salgisini arttiran glikokinaz aktivatörleridir.
申请公布号 TR200102805(T2) 申请公布日期 2002.04.22
申请号 TR20010002805T 申请日期 2000.03.20
申请人 F.HOFFMANN-LA ROCHE AG 发明人 THOMAS FRED BIZZARRO;LEA WENDY CORBETT;ANTONINO FOCELLA;FRANCIS JOSEPH GRIPPO;NANCY-ELLEN HAYNES;WILLIAM GEORGE HOLLAND;FRANCIS ROBERT KESTER;E.PAIGE MAHANEY;RAMAKANTH SARABU
分类号 A61K31/17;A61K31/4168;A61K31/42;A61K31/421;A61K31/426;A61K31/433;A61K31/4402;A61K31/455;A61K31/50;A61K31/505;A61P3/10;A61P43/00;C07C275/50;C07C317/44;C07C323/60;C07C323/62;C07D;C07D213/75;C07D213/80;C07D213/803;C07D213/82;C07D233/88;C07D237/20;C07D237/22;C07D239/42;C07D241/28;C07D253/07;C07D261/14;C07D263/34;C07D263/48;C07D277/20;C07D277/38;C07D277/46;C07D277/56;C07D277/58;C07D285/12;C07D285/135;(IPC1-7):C07D277/46;C07D80 主分类号 A61K31/17
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