发明名称 USE OF CHLOROQUINE, HYDROXY CHLOROQUINE AND 4 AMINO-QUINOLINIC DERIVATIVES TO OBTAIN A DRUG FOR THE ANTI RETROVIRAL THERAPY, ACTIVE TOWARDS HIV SENSITIVE STRAINS AND TOWARDS HIV STRAINS WHICH ARE RESISTANT TO BOTH NUCLEOSIDIC AND NONNUCLEOSIDIC REVERSE TRANSCRIPTASE INHIBITORS AND TO PROTEASES INHIBITORS
摘要 Use of at least one 4 amino-quinolinic derivative to obtain a drug for the anti-retroviral therapy, especially in the therapy of the HIV disease-infection caused by retroviral strains, which are sensitive and/or resistant to known therapies. Said 4 amino-quinolinic derivative is chloroquine and/or hydroxychloroquine and the drug can be orally administered once or several times a day.
申请公布号 CA2433237(A1) 申请公布日期 2003.12.28
申请号 CA20032433237 申请日期 2003.06.25
申请人 VALPHARMA S.A. 发明人 ALIGHIERI, TIZIANO;AVANESSIAN, SEROZH;VALDUCCI, ROBERTO
分类号 C07D215/46;A61K31/4706;A61P31/14;A61P31/18;A61P43/00;(IPC1-7):A61K31/470;A61K31/47;A61P31/12 主分类号 C07D215/46
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