发明名称 |
SMALL MOLECULE MODULATORS OF PCSK9 AND METHODS OF USE THEREOF |
摘要 |
A compound of Formula (I): or a pharmaceutically acceptable salt, hydrate, solvate, or racemic mixture or stereoisomer thereof, and methods for preventing or treating an LDL-cholesterol-related disease or disorder using such compound(s), and kits and compositions comprising such compound(s). |
申请公布号 |
EP2961765(A4) |
申请公布日期 |
2016.11.09 |
申请号 |
EP20140765405 |
申请日期 |
2014.03.14 |
申请人 |
ADAERATA, LIMITED PARTNERSHIP;AMORCHEM HOLDINGS INC. |
发明人 |
GUAY, DANIEL;CRANE, SHELDON;LACHANCE, NICOLAS;CHIASSON, JEAN-FRANÇOIS;TRUONG, VOUY LINH;LACOMBE, PATRICK;SKOREY, KATHRYN;SEIDAH, NABIL G. |
分类号 |
C07K5/083;A61K38/06;A61P3/06;C07K5/027;C07K5/08 |
主分类号 |
C07K5/083 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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