发明名称 SMALL MOLECULE MODULATORS OF PCSK9 AND METHODS OF USE THEREOF
摘要 A compound of Formula (I): or a pharmaceutically acceptable salt, hydrate, solvate, or racemic mixture or stereoisomer thereof, and methods for preventing or treating an LDL-cholesterol-related disease or disorder using such compound(s), and kits and compositions comprising such compound(s).
申请公布号 EP2961765(A4) 申请公布日期 2016.11.09
申请号 EP20140765405 申请日期 2014.03.14
申请人 ADAERATA, LIMITED PARTNERSHIP;AMORCHEM HOLDINGS INC. 发明人 GUAY, DANIEL;CRANE, SHELDON;LACHANCE, NICOLAS;CHIASSON, JEAN-FRANÇOIS;TRUONG, VOUY LINH;LACOMBE, PATRICK;SKOREY, KATHRYN;SEIDAH, NABIL G.
分类号 C07K5/083;A61K38/06;A61P3/06;C07K5/027;C07K5/08 主分类号 C07K5/083
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