发明名称 METHOD FOR PREPARING 17A-ETHINYL-17B-HYDROXY-18-METHYL-4,15-ESTRADIEN-3-ON AND THE NOVEL STARTING COMPOUNDS FOR THIS METHOD
摘要 A process and novel starting materials for the production of 17 alpha -ethynyl-17 beta -hydroxy-18-methyl-4,15-estradien-3-one of Formula I <IMAGE> (I) are disclosed. Novel 17-ketone starting materials have the Formula II <IMAGE> (II) wherein R is an alkyl residue of 1-3 carbon atoms and <IMAGE> is the grouping <IMAGE> wherein R' is an acyl group of up to 10 carbon atoms.
申请公布号 GR861126(B) 申请公布日期 1986.09.30
申请号 GR19860101126 申请日期 1986.04.29
申请人 SCHERING AG 发明人 DR. HOFMEISTER HELMUT;DR. LAURENT HENRY;DR. LORENZ HANS-PETER;DR. WIECHERT RUDOLF
分类号 A61K31/565;C07J1/00;C07J7/00;C07J75/00 主分类号 A61K31/565
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