发明名称 CRYSTALLINE SOLVATES AND COMPLEXES OF (1S)-1,5-ANHYDRO-1-C-(3-((PHENYL)METHYL)PHENYL)-D-GLUCITOL DERIVATIVES WITH AMINO ACIDS AS SGLT2 INHIBITORS FOR THE TREATMENT OF DIABETES
摘要 The present invention relates to physical crystal structures of a compound of the formula I: wherein R1, R2, R2a, R3 and R4 are as defined herein, especially pharmaceutical compositions containing structures of compound I or II, processes for preparing same, intermediates used in preparing same, and methods of treating diseases such as diabetes using such structures.
申请公布号 KR20090023643(A) 申请公布日期 2009.03.05
申请号 KR20087031643 申请日期 2007.06.21
申请人 BRISTOL-MYERS SQUIBB COMPANY 发明人 GOUGOUTAS JACK Z.;LOBINGER HILDEGARD;RAMAKRISHNAN SRIVIDYA;DESHPANDE PRASHANT P.;BIEN JEFFREY T.;LAI CHIAJEN;WANG CHENCHI;RIEBEL PETER;GROSSO JOHN ANTHONY;NIRSCHL ALEXANDRA A.;SINGH JANAK;DIMARCO JOHN D.
分类号 C07D309/10;A61K31/70;A61P3/10 主分类号 C07D309/10
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