发明名称 2-(R-THIO)-10-[3-(4-R-PIPERAZINE-1-YL)PROPYL]-10H-PHENOTHIAZINE FOR TREATING A BETA-AMYLOIDOSES OR ALPHA-SYNUCLEOPATHY AND METHOD FOR DIAGNOSIS OR PREDIAGNOSIS THEREOF
摘要 FIELD: medicine.SUBSTANCE: invention relates to use of 2-(R-thio)-10-[3-(4-R-piperazin-1-yl)propyl]-10H-phenothiazine according to general formula I for treating a β-amyloidopathy or α-synucle- opathy followed by a cerebral protein deposit and reduced activity of cerebral ABCC1-transporter, including Alzheimer's dementia, Parkinson's disease or Lewy body dementia. According to general formula I R- Methyl group, R- Ethyl group, R- Hydrogen and R- Hydrogen.EFFECT: treatment of β-amyloidopathy or α-synucleopathy.3 cl, 12 dwg
申请公布号 RU2587154(C2) 申请公布日期 2016.06.20
申请号 RU20130110018 申请日期 2011.08.30
申请人 IMMUNGENETIKS AG 发明人 PANKE JENS
分类号 C07D417/06;A61K31/5415;A61P25/28;C07D417/14 主分类号 C07D417/06
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