发明名称 |
Estrogen agonists/antagonists. |
摘要 |
Compounds of formula A inhibit bone resorption and bone turnover, prevent bone loss, preserve bone strength and decrease serum cholesterol without causing prostate hypertrophy in male mammals: <CHEM> and E and B are selected from CH and N. R<4> is H, OH, F or Cl.e |
申请公布号 |
ZA9905029(B) |
申请公布日期 |
2001.02.05 |
申请号 |
ZA19990005029 |
申请日期 |
1999.08.05 |
申请人 |
PFIZER PRODUCTS INC. |
发明人 |
KIMBERLY O'KEEFE CAMERON;PAUL ANDREW DASILVA-JARDINE;ROBERT LOUIS ROSATI;HUA ZHU KE |
分类号 |
C07D295/08;A61K31/40;A61K31/435;A61K31/44;A61K31/4427;A61K31/4439;A61K31/445;A61K31/4453;A61K31/47;A61K31/472;A61K31/4725;A61P3/04;A61P3/06;A61P5/32;A61P19/10;C07D217/24;C07D401/12 |
主分类号 |
C07D295/08 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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