| 发明名称 |
DERIVATIVES OF N-SULFONYL-2-OXOINDOLE, METHOD OF THEIR SYNTHESIS, INTERMEDIATE COMPOUNDS AND PHARMACEUTICAL COMPOSITION CONTAINING AGENT THAT SHOWS ACTIVITY WITH RESPECT TO VASOPRESSIN AND/OR OXYTOCIN RECEPTORS |
| 摘要 |
FIELD: organic chemistry. SUBSTANCE: invention describes derivatives of N-sulfonyl-2- -oxoindole of the general formula (I) <EMI ID=0.282 HE=48 WI=42 TI=CHI> where values R<SB>1</SB>-R<SB>6</SB> and m are given in point 1 of the invention. It describes also a method of their synthesis, intermediate substances and a pharmaceutical compositions based on compounds of the formula (I) showing affinity to vasopressin and/or oxytocin receptors. EFFECT: improved method of synthesis, affinity to receptors. 19 cl, 7 tbl, 211 ex
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| 申请公布号 |
RU2135469(C1) |
申请公布日期 |
1999.08.27 |
| 申请号 |
RU19930055882 |
申请日期 |
1993.01.28 |
| 申请人 |
ELF SANOFI |
发明人 |
LOIS FULON;ZHORZH GAREIA;DINO NIZATO;RISHAR RU;KLODIN SERRADEJL'-LEGAL';ZHERAR VALETT;ZHAN VAN'ON |
| 分类号 |
A61K31/40;A61K31/403;A61K31/404;A61P9/02;A61P43/00;C07C309/86;C07C309/87;C07C323/66;C07D;C07D209/32;C07D209/34;C07D209/92;C07D209/96;C07D401/12;C07D403/12;C07D405/12;C07D405/14;C07D409/12;C07D471/10;C07D491/10;C07D491/107;C07D495/10;(IPC1-7):C07D209/96 |
主分类号 |
A61K31/40 |
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