发明名称 Phenyloxadiazole derivatives as PGDS inhibitors
摘要 This invention is directed to a compound of formula (I):; wherein R1, R2 and R3 are as defined herein, a pharmaceutical composition comprising the compound, intermediates and processes for making said compounds, and the use of the compound to treat allergic and/or inflammatory disorders, particularly disorders such as allergic rhinitis, asthma, chronic obstructive pulmonary disease (COPD) and age-related macular degeneration (AMD).
申请公布号 US9469627(B2) 申请公布日期 2016.10.18
申请号 US201213439511 申请日期 2012.04.04
申请人 Sanofi 发明人 Vandeusen Christopher L.;Weiberth Franz J.;Gill Harpal S.;Lee George;Hillegass Andrea
分类号 C07D413/14;A61K31/506;C07D271/06 主分类号 C07D413/14
代理机构 Cooley LLP 代理人 Cooley LLP
主权项 1. A compound of formula (I): wherein R1 is hydrogen or C1-C6 alkyl; R2 is hydrogen, halogen or C1-C3 alkyl; and R3 is hydroxyalkyl.
地址 Paris FR