| 发明名称 |
Improved oxidation process with enhanced safety and use thereof |
| 摘要 |
<p>The present invention provides a safe and effective process for the selective oxidation of a 5-O-protected-LLF-28249-alpha compound to the corresponding 23-keto compound of formula I wherein R is a protecting group. The present invention also provides the use of the selective oxidation process in the manufacture of moxidectin.</p> |
| 申请公布号 |
AU2006203353(B8) |
申请公布日期 |
2007.12.13 |
| 申请号 |
AU20060203353 |
申请日期 |
2006.08.04 |
| 申请人 |
WYETH |
发明人 |
JIGNESH PATEL;PASQUALE MASSARA;STEFANIA SAPIENZA;MARCO CARACO;GIUSEPPE MIRAGLIA |
| 分类号 |
C07D493/22 |
主分类号 |
C07D493/22 |
| 代理机构 |
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代理人 |
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| 主权项 |
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| 地址 |
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