Combined preparations, containing 1,4-benzothiepine-1,1-dioxide derivatives and other active substances, and the use thereof.

摘要

A composition comprises a benzothiepin-1,1-dioxide derivative (I) or its salt or functional derivative and another active agent (II). A composition comprises a benzothiepin-1,1-dioxide derivative of formula (I) or its salt or functional derivative and another active agent (II). R<1>, R<4> and R<5> = methyl, ethyl, propyl or butyl; R<2> = hydrogen, hydroxy or (1-6C alkyl)amino; R<3> = mono- to tetra-saccharide residue, or the residue of a mono- to tetra-amino acid, all optionally substituted one or more times by protecting groups; Z = (CO)n-(0-16C)alkyl, (CO)n-(0-16C)alkylamino, (CO)n(0-16C)alkoxy, (CO)n(1-16C)alkyl-(CO)m or bond; and n and m = 0 or 1.