发明名称 SUBSTITUTED ALKYLAMINE DERIVATIVES AND METHODS OF USE
摘要 Selected heterocyclic compounds are effective for prophylaxis and treatment of diseases, such as angiogenesis mediated diseases. The invention encompasses novel compounds, analogs, prodrugs and pharmaceutically acceptable derivatives thereof, pharmaceutical compositions and methods for prophylaxis and treatment of diseases and other maladies or conditions involving, cancer and the like. The subject invention also relates to processes for making such compounds as well as to intermediates useful in such processes.
申请公布号 EA006973(B1) 申请公布日期 2006.06.30
申请号 EA20030000788 申请日期 2002.01.11
申请人 AMGEN INC. 发明人 CHEN GUOQING;ADAMS JEFFREY;BEMIS JEAN;BOOKER SHON;CAI GUOLIN;CROGHAN MICHAEL;DIPIETRO LUCIAN;DOMINGUEZ CELIA;ELBAUM DANIEL;GERMAIN JULIE;GEUNS-MEYER STEPHANIE;HANDLEY MICHAEL;HUANG QI;KIM JOSEPH, L.;KIM TAE-SEONG;KISELYOV ALEXANDER;OUYANG XIAOHU;PATEL VINOD, F.;SMITH LEON, M.;STEC MARKIAN;TASKER ANDREW;XI NING;XU SHIMIN;YYAN CHESTER, CHENGUANG
分类号 C07D409/12;A61K31/4436;A61K31/444;A61K31/4709;A61K31/496;A61K31/501;A61K31/506;A61K31/5377;A61P9/10;A61P11/06;A61P15/08;A61P17/06;A61P27/02;A61P29/00;A61P35/00;A61P43/00;C07D213/82;C07D401/12;C07D401/14;C07D405/12;C07D405/14;C07D407/14;C07D409/04;C07D409/14;C07D413/14;C07D417/14;C07D471/04 主分类号 C07D409/12
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