发明名称 |
HETEROARYL SUBSTITUTED PYRROLO[2,3-b]PYRIDINES AND PYRROLO[2,3-b]PYRIMIDINES AS JANUS KINASE INHIBITORS |
摘要 |
The present invention provides heteroaryl substituted pyrrolo[2,3-b]pyridines and heteroaryl substituted pyrrolo[2,3-b]pyrimidines that modulate the activity of Janus kinases and are useful in the treatment of diseases related to activity of Janus kinases including, for example, immune-related diseases, skin disorders, myeloid proliferative disorders, cancer, and other diseases. |
申请公布号 |
US2010022522(A1) |
申请公布日期 |
2010.01.28 |
申请号 |
US20090549170 |
申请日期 |
2009.08.27 |
申请人 |
INCYTE CORPORATIONN, A DELAWARE CORPORATION |
发明人 |
RODGERS JAMES D.;SHEPARD STACEY;MADUSKUIE, JR. THOMAS P.;WANG HAISHENG;FALAHATPISHEH NIKOO;RAFALSKI MARIA;ARVANITIS ARGYRIOS G.;STORACE LOUIS;JALLURI RAVIKUMAR;FRIDMAN JORDAN S.;VADDI KRISHNA |
分类号 |
A61K31/437;A61K31/506;A61K31/519;A61K31/5377;A61K31/541;A61P17/00;A61P29/00;A61P31/12;A61P35/00;A61P37/06;C07D401/14;C07D413/14;C07D417/14;C07D471/04;C07D487/04 |
主分类号 |
A61K31/437 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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