| 发明名称 |
A PROCESS FOR THE PREPARATION OF TOFACITINIB CITRATE |
| 摘要 |
The present invention provides a process for the preparation of tofacitinib citrate of Formula I. Specifically, the present invention provides an enzymatic route for the preparation of tofacitinib of Formula II, which is converted to tofacitinib citrate of Formula I. |
| 申请公布号 |
WO2016132341(A1) |
申请公布日期 |
2016.08.25 |
| 申请号 |
WO2016IB50946 |
申请日期 |
2016.02.22 |
| 申请人 |
SUN PHARMACEUTICAL INDUSTRIES LIMITED |
发明人 |
BHANDYA, Somashekar Rudrappa;MADHRA, Mukesh Kumar |
| 分类号 |
C07D487/04;A61K31/519 |
主分类号 |
C07D487/04 |
| 代理机构 |
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