发明名称 PYRANONE COMPOUNDS FOR TREATMENT OF RETROVIRAL INFECTION
摘要 The present invention relates to compounds of formula I and II which are pyran-2-ones, 5,6-dihydro-pyran-2-ones, 4-hydroxy-benzopyran-2-ones, 4-hydroxy-cycloalkyl[b]pyran-2-ones, and derivatives thereof, useful for inhibiting a retrovirus in a mammalian cell infected with said retrovirus.wherein R10 and R20 taken together are:
申请公布号 NZ285510(A) 申请公布日期 1998.03.25
申请号 NZ19950285510 申请日期 1995.05.04
申请人 PHARMACIA & UPJOHN CO 发明人 ROMINES, KAREN RENE;BUNDY, GORDON L;SCHWARTZ, THERESA M;TOMMASI, RUBEN A;STROHBACH, JOSEPH WALTER;TURNER, STEVEN RONALD;JOHNSON, PAUL D;SKULNICK, HARVEY IRVING;SKALETZKI, LOUIS L;ANDERSON, DAVID JOHN;MORRIS, JOEL;GAMMILL, RONALD B;LUKE, GEORGE P;THAISRIVONGS, SUVIT;ARISTOFF, PAUL ADRIAN
分类号 A61K31/365;A61K31/366;A61K31/415;A61K31/425;A61K31/44;A61K31/4427;A61K31/443;A61K31/47;A61K31/4709;A61K31/505;A61K31/506;A61K31/54;A61P31/12;C07D;C07D309/32;C07D309/38;C07D309/40;C07D311/02;C07D311/08;C07D311/74;C07D311/94;C07D401/12;C07D403/12;C07D405/00;C07D405/12;C07D405/14;C07D407/00;C07D409/00;C07D417/00;C07D417/12;(IPC1-7):C07D309/32 主分类号 A61K31/365
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