发明名称 4-ARYLMETHYLOXYMETHYL PIPERIDINE ALS TACHYKININ ANTAGONISTEN
摘要 PCT No. PCT/GB93/02214 Sec. 371 Date Apr. 13, 1995 Sec. 102(e) Date Apr. 13, 1995 PCT Filed Oct. 27, 1993 PCT Pub. No. WO94/10165 PCT Pub. Date May 11, 1994The present invention is directed to compounds of the formula (I) <IMAGE> wherein R1, R2, R3, R4, R5, R6, and R7 are defined herein, and pharmaceutically acceptable salts thereof, which are useful as tachykinin antagonists,
申请公布号 DE69327541(D1) 申请公布日期 2000.02.10
申请号 DE1993627541 申请日期 1993.10.27
申请人 MERCK SHARP & DOHME LTD., HODDESDON 发明人 HARRISON, TIMOTHY;MACLEOD, ANGUS MURRAY;STEVENSON, GRAEME IRVINE;WILLIAMS, BRIAN JOHN
分类号 C07D211/20;A61K31/40;A61K31/44;A61K31/4427;A61K31/445;A61K31/4465;A61K31/451;A61P1/00;A61P1/08;A61P9/00;A61P11/00;A61P13/02;A61P15/00;A61P25/02;A61P25/04;A61P25/06;A61P25/08;A61P25/18;A61P25/20;A61P25/24;A61P25/26;A61P25/28;A61P25/30;A61P29/00;A61P35/00;A61P37/00;A61P37/08;A61P43/00;C07D207/08;C07D211/22;C07D211/96;C07D213/40;C07D401/06;C07D401/12;C07D413/06;C07D417/06;C07D521/00;(IPC1-7):C07D401/06 主分类号 C07D211/20
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