发明名称 Nitric oxide synthase inhibitors derived from cyclic amidines
摘要 Compounds having formula (I) wherein R<1>, R<5>, R<6> and R<7> are hydrogen or certain specified substituents; R<8> and R<9> are independently hydrogen, hydroxy or alkoxy; and X, A and B are independently NR<2>, O, S, SO, SO2, CH=CH or (CH2)p, p being 0-6; are useful as nitric oxide synthase inhibitors.
申请公布号 ZA9603742(B) 申请公布日期 1997.07.09
申请号 ZA19960003742 申请日期 1996.05.10
申请人 G.D. SEARLE & CO. 发明人 HANSEN, DONALD, W., JR.;TIMOTHY J. HAGEN;STEVEN W. KRAMER;SUZANNE METZ;KAREN B. PETERSON;DALE P. SPANGLER;MIHALY V. TOTH;KAM F. FOK;KEITH R. WEBBER;FOE S. TJOENG;BARNETT S. PITZELE
分类号 A61K31/00;A61K31/40;A61K31/445;A61K31/55;A61P9/00;A61P9/02;A61P31/00;A61P37/00;A61P37/06;C07D207/22;C07D207/24;C07D211/72;C07D211/74;C07D223/12;C07D243/08;C07D267/08;C07D267/10;C07D403/06;C07D413/06;C07D413/12;C07D471/10 主分类号 A61K31/00
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